Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_07109
Ion Channel
Neuronal acetylcholine receptor subunit alpha9/alpha10
Peptide Function
Antagonist
Gene Name
CHRNA9/CHRNA10
Activity Data (nM)
IC50
0.36 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
GCXTDPRCRXXCXK
Peptide UniProt Accession
Not available
UniParc
Not available
Peptide Synonyms/Alias
Not available
Peptide Species
Conus snails
Peptide Name
Not available
CAS Number
Not available
Experimental Conditions
pH
pH 7.2–7.5
Holding Potential (mV)
−70 mV
Temperature
21−24 °C
Test Method
Patch-clamping
Test Species
Xenopus Oocyte
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
nAChRs
Ion Channel UniProt Accession
Source Organism
Homo sapiens (Human)
References & Disease Information
Disease
Not specified
PubChem CID
URL
Not available
PMID
Patent
Not available